Benzothiazole and benzimidazole derivatives and antiulcer agent

Details Benzothiazole and benzimidazole derivatives and antiulcer agent Benzothiazole and benzimidazole derivatives and antiulcer agent

1993-03-25

1994-03-15

Gerstl, Robert

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

514395, 548166, 548169, 5483071, C07D23528, C07D27776, A61K 31415, A61K 31425

Patent

active

052946290

ABSTRACT:
A novel benzothiazole or benzimidazole derivative represented by formula (I) ##STR1## wherein X represents a sulfur atom or a NH group; R.sup.1 represents a hydrogen atom, a lower alkoxy group, a chlorine atom, a bromine atom or an iodine atom; R.sup.2 represents a hydrogen atom a substituted or unsubstituted lower alkyl group, a vinyl group, an aryl group or an acyl group; m is an integer of 1, 2 or 3; and n is an integer of 0, 1 or 2, which shows an excellent acid secretion suppressing effect and gastric mucosa protecting effect, and an antiulcer agent containing the same as an active ingredient.

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