Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...
Patent
1996-05-31
1998-06-02
Shah, Mukund J.
Organic compounds -- part of the class 532-570 series
Organic compounds
Heterocyclic carbon compounds containing a hetero ring...
514415, 514418, 514419, 548483, 548484, 548485, 548486, 548495, C07D20902, C07D20942, A61K 3140
Patent
active
057602484
ABSTRACT:
A description is given of tachykinin receptor antagonists having general formula (I) ##STR1## their preparation and use in pharmaceutical formulations.
REFERENCES:
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Mantyh et al., Proc. Natl. Acad. Sci. USA, 85, 3235 (1988).
STN search report for: Potier et al., New NK-1 Tachykinin Receptor Antagonists Based on a Alicyclic Amino Acids as a Template: Stereoselective Synthesis and Chirality Investigation by NMR, Pept. 1994, Proc. Eur. Symp., 23rd, Meeting Date 1994, p. 315-, 1995.
Sisto et al., Synthesis and Biological Evaluation of Novel NK-1 Tachykinin Receptor Antagonists: The Use of Cycloalkyl Amino Acids as a Template, Biopolymers, vol. 36, No. 4, pp. 511-524, Oct. 1995.
Peters et al., Amer. Rev. Resp. Dis. 145,835 (1992).
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Arcamone Federico
Fincham Christopher
Lombardi Paolo
Manzini Stefano
Potier Edoardo
A.Menarini Industrie Farmaceutiche Riunite S.r.l.
Coleman Brenda
Shah Mukund J.
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