Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...
Reexamination Certificate
2005-07-25
2008-12-30
Shameem, Golam M (Department: 1626)
Organic compounds -- part of the class 532-570 series
Organic compounds
Heterocyclic carbon compounds containing a hetero ring...
C548S300100, C548S301700, C548S302700, C544S106000, C544S111000, C544S132000, C544S358000
Reexamination Certificate
active
07470795
ABSTRACT:
Disclosed is a multi-step process for preparing a compound of Formula I:wherein R1to R3are as defined herein. The compounds of formula I inhibit the binding of human intercellular adhesion molecules to the Leukointegrins. As a result, these compounds are useful in the treatment of inflammatory and immune cell-mediated diseases.
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Frutos Rogelio Perez
Krishnamurthy Dhileepkumar
Kroeber Jutta
Nicola Thomas
Nummy Laurence John
Boehringer Ingelheim International GmbH
Boehringer Ingelheim Pharmaceuticals Inc.
Datlow Philip I.
Devlin Mary-Ellen M.
Morris Michael P.
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