Substituted benzyl ester derivative and use thereof

Details Substituted benzyl ester derivative and use thereof Substituted benzyl ester derivative and use thereof

2011-07-19

2011-07-19

Oh, Victor (Department: 1625)

Food or edible material: processes, compositions, and products

Products per se, or processes of preparing or treating...

Nutritional or dietetic supplement, including table salt

C514S544000, C549S434000, C549S445000, C549S447000

Reexamination Certificate

active

07981460

ABSTRACT:
The present invention relates to a pharmaceutical composition, a food composition or a cosmetic composition, containing one or more kinds of a compound represented by the following formula (I′)wherein R1 is a hydrogen atom, a hydroxyl group, a methoxy group or an ethoxy group, R2 is a hydroxyl group, a methoxy group or an acetoxy group, or R1 and R2 in combination optionally form a methylenedioxy group,R is represented by the following formulawherein Y is an ethylene group or a vinylene group, m and n are each an integer of 0 to 7, which satisfy m+n=2 to 8, and R3 and R4 are each independently a hydrogen atom, a methyl group or an ethyl group,provided that,(1) when R1 is a methoxy group, then R2 is not a hydroxyl group; and(2) when R1 is a hydroxyl group, then R2 is not a hydroxyl group and an acetoxy group.According to the present invention, a stable capsinoid derivative is provided, and a pharmaceutical composition, a food composition, a cosmetic composition and the like containing the derivative as an active ingredient can be provided.

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