Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Patent
1999-10-15
2000-11-21
Stockton, Laura L.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
5483751, 5483771, A61K 31415, C07D23116
Patent
active
061503932
ABSTRACT:
Disclosed herein are non-endogenous, constitutively activated forms of the human 5-HT.sub.2A and human 5-HT.sub.2C receptors and uses of such receptors to screen candidate compounds. Further disclosed herein are candidate compounds identified by the screening method which act at the 5HT.sub.2A receptors. Yet further disclosed is a new class of compounds which act at the 5HT.sub.2A receptors.
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Beeley Nigel R. A.
Behan Dominic P.
Chalmers Derek T.
Foster Richard J.
Glen Robert C.
Arena Pharmaceuticals Inc.
Stockton Laura L.
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