Saccharin derivatives useful as proteolytic enzyme inhibitors an

Details Saccharin derivatives useful as proteolytic enzyme inhibitors an Saccharin derivatives useful as proteolytic enzyme inhibitors an

1991-11-15

1993-08-17

Higel, Floyd D.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Heterocyclic carbon compounds containing a hetero ring...

514338, 514373, 548210, A61K 3141

Patent

active

052369170

ABSTRACT:
Novel 2-substituted saccharins which inhibit the enzymatic activity of proteolytic enzymes, are useful in the treatment of degenerative diseases and have the formula ##STR1## wherein: L is --O--, --S--, --SO-- or --SO.sub.2 --;

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