Pyrazolo [1,5-a] pyrimidine derivative and nad (p) h oxidase...

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

Reexamination Certificate

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Details

C544S281000

Reexamination Certificate

active

07662826

ABSTRACT:
A compound represented by the formula (Ia) (wherein R1a, R2a, and R3 to R5 are the same as defined in the description), a prodrug thereof, a pharmaceutically acceptable salt thereof, or solvate thereof. The compounds are useful in the prevention of or treatment for diseases relating to NAD(P)H.

REFERENCES:
patent: 4081545 (1978-03-01), Clayton
patent: 4166817 (1979-09-01), Ferres et al.
patent: 4918074 (1990-04-01), Tsuda et al.
patent: 4992442 (1991-02-01), Tsujitani et al.
patent: 5420128 (1995-05-01), Kiyokawa et al.
patent: 5478838 (1995-12-01), Arita et al.
patent: 5888941 (1999-03-01), Bartroli et al.
patent: 6229011 (2001-05-01), Chen et al.
patent: 2001/0025047 (2001-09-01), Levin et al.
patent: 2001/0046989 (2001-11-01), Levin et al.
patent: 2002/0132826 (2002-09-01), Levin et al.
patent: 1 568 962 (1980-06-01), None
patent: 1 579 362 (1980-11-01), None
patent: 06-009638 (1994-01-01), None
patent: 07-242670 (1995-09-01), None
patent: 07-267960 (1995-10-01), None
patent: 10-120683 (1998-05-01), None
patent: 2001-302666 (2001-10-01), None
patent: WO 99/10313 (1999-03-01), None
patent: WO 99/18076 (1999-04-01), None
patent: WO 99/59526 (1999-11-01), None
patent: WO 01/90101 (2001-11-01), None
patent: WO 02/24613 (2002-03-01), None
patent: WO 02/28820 (2002-04-01), None
Bartroli et al., “New Azole Antifungals. 2. Synthesis and Antifungal Activity of Heterocyclecarboxamide Derivatives of 3-Amino-2-aryl-1-azolyl-2-butanol,”J. Med. Chem., 41:1855-1868 (1998).
Checchi et al., “5-Aminopyrazole derivatives. III. Acids of pyrazopyrimidine, pyrazopyridone, pyrazopyridine, and some derivatives,”Gazzetta Chimica Italiana, 86:631-645 (1956) (with attached English-language abstract).
Checchi et al., “Derivaties of 5-aminopyrazole. IV. Synthesis of heterocyclic derivatives,”Gazzetta Chimica Italiana, 87:597-614 (1957) (with attached English-language abstract).
Elworthy et al., “N-Arylpiperazinyl-N′-propylamino Derivatives of Heteroaryl Amides as Functional Uroselective α1-Adrenoceptor Antagonists,”J. Med. Chem., 40:2674-2687 (1997).
Mustazza et al., “Synthesis of Pyrazolo[1,5-a]-1,2,4-Triazolo[1,5-a]-and Imidazo[1,2-a]pyrimidines Related to Zaleplon, a New Drug for the Treatment of Insomnia,”J. Heterocyclic Chem., 38:1119-1129 (2001).
Novinson et al., “Synthesis and Antifungal Properties of Certain 7-Alkylaminopyrazolo[1,5-a]pyrimidines,”Journal of Medicinal Chemistry, 20(2):296-299 (1977).
Takamizawa et al., “Studies on Pyrimidine Derivatives and Related Compounds, LIX. Syntheses of 2,3- Dihydro-1H-pyrazolo[5,1-b]purin-2-ones,”Chem. Pharm. Bull., 16(11):2195-2199 (1968).

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