Process for making HIV protease inhibitors

Details Process for making HIV protease inhibitors Process for making HIV protease inhibitors

1995-06-07

1997-04-08

Bernhardt, Emily

Organic compounds -- part of the class 532-570 series

Organic compounds

Nitrogen attached directly or indirectly to the purine ring...

544137, 544360, 544364, 544373, 544374, 544390, 546146, 546147, 548217, 549552, C07D40906, C07D40914, C07D40506, C07D24104

Patent

active

056189397

ABSTRACT:
A process is disclosed for making a chiral compound of the formula ##STR1## comprising reacting an epoxide compound of the formula ##STR2## and an amide of the formula ##STR3## in the presence of a strong base at a low temperature.

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