Pro-prodrugs, their production and use

Details Pro-prodrugs, their production and use Pro-prodrugs, their production and use

1994-09-20

1999-03-02

Harrison, Robert M.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Carbohydrate doai

536 64, 536 187, 552201, A61K 4748

Patent

active

058771581

ABSTRACT:
Substrate-spacer-prodrug compounds (pro-prodrugs) suited for site specific delivery of drugs, a process of preparing them and their use are described.

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Bundgaerd "The Double Prodrug Concept and its Applications", Advanced Drug Delivery Reviews, 3, pp. 39-65, 1989.

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