Organic compounds -- part of the class 532-570 series – Organic compounds – Four or more ring nitrogens in the bicyclo ring system
Reexamination Certificate
2006-04-18
2006-04-18
McKenzie, Thomas C. (Department: 1624)
Organic compounds -- part of the class 532-570 series
Organic compounds
Four or more ring nitrogens in the bicyclo ring system
C544S278000
Reexamination Certificate
active
07030240
ABSTRACT:
The invention relates to 5-HT receptor antagonists. Novel piperidinylamino-thieno[2,3-d] pyrimidine compounds represented by Formula I, and synthesis and uses thereof for treating diseases mediated directly or indirectly by 5-HT receptors, are disclosed. Such conditions include central nervous system disorders such as anxiety, depression, schizophrenia, neural injury, stroke, and migraine. Methods of preparation and novel intermediates and pharmaceutical salts thereof are also included.
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International Search Report for PCTY/US04/09944, mailed Mar. 1, 2005.
Bar-Haim Shay
Becker Oren
Chen Dongli
Cheruku Srinivasa Rao
Dhanoa Dale S.
Elrifi Ivor R.
McKenzie Thomas C.
Mintz Levin Cohn Ferris Glovsky and Popeo P.C.
Predix Pharmaceuticals Holdings, Inc.
Triano, III Nicholas P.
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