Phosphonate and phosphinate pyrazolylamide glucokinase...

Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...

Reexamination Certificate

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C544S408000, C548S953000, C549S475000

Reexamination Certificate

active

07910747

ABSTRACT:
Pyrazoloamides are provided which are phosphonate and phosphinate glucokinase activators that are useful in treating diabetes and related diseases and have the structurewhereinis a pyrazoyl ring;R4is —(CH2)n—Z—(CH2)m—PO(OR7)(OR8),—(CH2)nZ—(CH2)m—PO(OR7)R9, or—(CH2)nZ—(CH2)m—PO(R9)(R10);R5and R6are independently selected from H, alkyl and halogen;Y is R3(CH2)s, wherein R3is aryl , s is 0, X is a bond; andn, Z, m, R4, R5, R6, and R7are as defined herein;or a pharmaceutically acceptable salt thereof.

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