Phosphinyloxy, oxime and carboxylic acid derivatives which...

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Peptide containing doai

Reexamination Certificate

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C514S018700, C514S019300, C514S063000, C514S089000, C514S277000, C514S340000, C514S345000, C514S352000, C514S357000, C546S192000, C546S210000, C546S248000, C548S253000, C558S012000, C558S166000, C560S015000, C530S331000

Reexamination Certificate

active

11293060

ABSTRACT:
The present invention relates to compounds of Formula I, and pharmaceutically acceptable salts or solvates thereof, or solvates of such salts,which compounds inhibit carboxypeptidase U and thus can be used in the prevention and treatment of diseases associated with carboxypeptidase U. In further aspects, the invention relates to compounds of the invention for use in therapy; to processes for preparation of such new compounds; to pharmaceutical compositions containing at least one compound of the invention, or a pharmaceutically acceptable salt or solvate thereof, as active ingredient; and to the use of the active compounds in the manufacture of medicaments for the medical use indicated above.

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