Partial and full agonists of A1 adenosine receptors

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Carbohydrate doai

Reexamination Certificate

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Details

C514S045000, C536S027100, C536S027130, C536S027200, C536S027210, C536S027300, C536S027620

Reexamination Certificate

active

10855471

ABSTRACT:
Disclosed are novel compounds that are partial and full A1adenosine receptor agonists, useful for treating various disease states, in particular tachycardia and atrial flutter, angina, and myocardial infarction.

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patent: WO 01/40243 (2001-06-01), None
Van Der Wenden, E. et al: “5′-Substituted adenosine analogs as new high-affinity partial agonists for the adenosine A1 receptor” J. Med Chem 1998, 41, pp. 102-108.
Tilburg, E. et al: “N6.5′-Disubstituted adenosine derivatives as partial agonists for the human adenosine A3 receptor”, J. Med Chem, 1999, 42, pp. 1393-1400.
Smejkal, R.M. et al: “Muscarinic receptor subtype specificity of 5′(isobutylthio)-adenosine (SIBA) and its analogues”, Gen Pharmac., 20(3) pp. 385-392, 1989.

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