Non-steroidal androgen receptor modulators, preparation...

Details Non-steroidal androgen receptor modulators, preparation... Non-steroidal androgen receptor modulators, preparation...

2006-05-26

2010-06-15

Desai, Rita J (Department: 1625)

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

C564S342000, C564S345000, C514S471000, C514S649000

Reexamination Certificate

active

07737288

ABSTRACT:
Non-steroidal androgen receptor modulating compounds of the general formula (I), their pharmaceutically acceptable salts, preparation process and pharmaceutically compositions containing the said compounds are disclosed. Such compounds of the general formula (I) or their pharmaceutically acceptable salts can be used for preparing non-steroidal medicines to treat and/or prevent conditions or diseases such as prostatic hyperplasia, prostate cancer, hirsutism, severe hormone-dependent alopecia or acne, etc. as a result of androgen receptor antagonistic activities.

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International Search Report for PCT/CN2006/001106 mailed Sep. 7, 2006.

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