Imidazoquinoline derivatives and their use as adenosine A3...

Details Imidazoquinoline derivatives and their use as adenosine A3... Imidazoquinoline derivatives and their use as adenosine A3...

2007-02-13

2007-02-13

Seaman, Margaret D. (Department: 1625)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

C546S084000

Reexamination Certificate

active

10499251

ABSTRACT:
The present invention relates to adenosine A3receptor ligands of the general formula (I), within those preferably antagonists, as well as their salts, solvates and isomers, and the pharmaceutical compositions containings them, to the use of the compounds of the general formula (I), as well as their salts, solvates and isomers, to the preparation of the compounds of the general formula (I) and their salts, solvates and isomers, furthermore to the new intermediates of the general formulae (II) and (III) and to the preparation thereof.

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Ager, Ian R. et al., J. Med. Chem., vol. 31(6), pp. 1098-1115 (1988).
Clements-Jewery, Stephen et al., J. Med. Chem., vol. 31(6), pp. 1220-1226 (1988).

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