Histamine H3 receptor ligands

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

Reexamination Certificate

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C548S569000, C548S570000

Reexamination Certificate

active

06878736

ABSTRACT:
Compounds of formula (I) (and pharmaceutically acceptable salts thereof) are histamine H3receptor ligands. A in the formula represents (CH2)m, m being from 1 to 3; B is (CH2)n, n being from 1 to 3; x is from 0 to 2; R1is C1to C10hydrocarbyl, in which up to 2 carbon atoms may be replaced by O, S or N; and up to 2 hydrogen atoms may be replaced by halogen; R2is H or C1to C15hydrocarbyl, in which up to 3 carbon atoms may be replaced by O, S or N, and up to 3 hydrogen atoms may be replaced by halogen; R3is absent when —Y—Z—R2is attached to W, or is H or C1to C7hydrocarbyl when —Y—Z—R2is not attached to W; W is nitrogen; X is —CH2—, —O— or —NR4—, R4being H or C1to C3alkyl; Y replaces a hydrogen atom on any of A, B, W and X, and is C2to C10alkylene, in which one non-terminal carbon atom may be replaced by O; and Z is (II), (III), (IV), (V), (VI), or (VII) wherein R5, R6and R7are independently H or C1to C15hydrocarbyl, in which up to 3 carbon atoms may be replaced by O or N, and up to 3 hydrogen atoms may be replaced by halogen, and Q is H or methyl, or Q is linked to R5or R7to form a five-membered ring or Q is linked to R2to form a six-membered ring

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