Fused ring dicationic anti-protozoan agents and their prodrugs

Organic compounds -- part of the class 532-570 series – Organic compounds – Amino nitrogen containing

Reexamination Certificate

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C564S229000, C564S238000, C546S106000, C546S306000, C560S008000, C560S034000, C514S297000, C514S357000, C514S533000, C514S534000, C514S633000, C514S634000

Reexamination Certificate

active

07825279

ABSTRACT:
Novel fused ring dicationic anti-protozoan compounds. Representative protozoan species include but are not limited toTrypanosoma brucei rhodesiense(T.b.r.) andPlasmodium falciparum. Prodrugs of these compounds can be used as an oral treatment for malaria and human African trypanosomiasis.

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