Fluoropyrrolidines as dipeptidyl peptidase inhibitors

Details Fluoropyrrolidines as dipeptidyl peptidase inhibitors Fluoropyrrolidines as dipeptidyl peptidase inhibitors

2007-02-27

2007-02-27

Powers, Fiona T. (Department: 1626)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

C514S321000, C514S326000, C514S343000, C514S422000, C514S423000, C546S125000, C546S198000, C546S208000, C546S279100, C548S518000, C548S530000, C548S540000

Reexamination Certificate

active

10481543

ABSTRACT:
The present invention relates to novel compounds, their use for inhibiting post prolin/analine-cleaving proteases, such as serine proteases, such as dipeptidyl peptidases, such as dipeptidyl peptidase IV (DPP-IV), and to methods for their production and their therapeutic utility.

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