Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Patent
1995-06-07
1997-05-20
Tsang, Cecilia
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
514218, 544361, 544368, 540575, A61K 31495, A61K 3155, C07D40100, C07D41900
Patent
active
056312571
ABSTRACT:
A benzoxazole derivative of the formula (1) or (2) which has an alicyclic diamine group at the 2-position: ##STR1## wherein R.sup.1, R.sup.2, R.sup.3, R.sup.4, R.sup.5, R.sup.6, X.sup.-, m and n are defined herein. The compound shows excellent 5-HT.sub.3 receptor antagonism and is useful as an antiemetic agent, a peristalsis controlling agent, an analgesic agent, an antianxiety agent and a schizophrenia treating agent.
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Amano Kazuko
Inoye Shigeharu
Iwamatsu Katsuyoshi
Izumi Masaaki
Konno Fukio
Koichi Shudo
Meiji Seika Kaisha Ltd.
Tsang Cecilia
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