Chemistry: natural resins or derivatives; peptides or proteins; – Peptides of 3 to 100 amino acid residues – Peptides with at least one nonpeptide bond other than a...
Patent
1988-12-13
1989-08-01
Foelak, Morton
Chemistry: natural resins or derivatives; peptides or proteins;
Peptides of 3 to 100 amino acid residues
Peptides with at least one nonpeptide bond other than a...
544106, 544159, 544176, 548336, 560126, 560129, C07C10350, C07D23364, C07D41312
Patent
active
048534633
ABSTRACT:
Novel amino acid derivatives useful as a therapeutic agent are disclosed. These amino acid derivatives and the pharmaceutically acceptable salts thereof have a human renin inhibitory effect when administered orally and are useful for treatment of hypertension, especially renin-associated hypertension.
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Akahane Kenji
Iizuka Kinji
Kamijo Tetsuhide
Kiso Yoshiaki
Kubota Tetsuhiro
Foelak Morton
Kissei Pharmaceutical Co. Ltd.
Nutter Nathan M.
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