Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...
Patent
1995-01-25
1997-10-21
Cooney, Jr., John M.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Heterocyclic carbon compounds containing a hetero ring...
514213, 514214, 514215, 514217, 514218, 514219, 514220, 514221, 514279, 514299, 514359, 514438, 514439, 514443, 514444, 514448, 540521, 540522, 546 38, A61K 3155, C07D49506
Patent
active
056796714
ABSTRACT:
The present invention relates to an amino acid derivative having an angiotensin I-converting enzyme inhibition activity, a vasopressin antagonism and an atrial natriuretic peptide hydrolase inhibition activity.
This amino acid derivative is represented by the following general formula (I): ##STR1## wherein R.sup.1 represents a hydrogen atom or an acyl group; R.sup.2 represents a hydrogen atom, a lower alkyl group, a cycloalkyl group, an ary group which may have a substituent, a heteroaryl group which may have a substituent, an arylalkyl group which may have a substituent or a heteroarylalkyl group which may have a substituent;
REFERENCES:
patent: 5238932 (1993-08-01), Flynn et al.
Flynn et al., J. Med. Chem., 36(16), pp. 2420-2423 (Aug. 1993).
Hayashi Kenji
Kotake Makoto
Matsuoka Toshiyuki
Miyake Kazutoshi
Mori Nobuyuki
Cooney Jr. John M.
Eisai Co. Ltd.
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