Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Patent
1988-06-08
1990-05-29
Brust, Joseph Paul
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
548540, C07C20708, A61K 3140
Patent
active
049296337
ABSTRACT:
As new compounds are provided a class of derivatives of actinonin represented by the general formula ##STR1## where R is a hydrogen or a lower alkyl group, which can exhibit the enzyme-inhibitory activities to a limited range of peptidases and show a remarkable enzyme-specificity, and which are effective to treat a cycloheximide-induced experimental amnesia in mice and are expectable to be useful to treat an amnesia in a mammalian animal, including human.
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Aoyagi Takaaki
Hachisu Mitsugu
Kondo Shin-ichi
Matsuhashi Yuji
Shibahara Seiji
Brust Joseph Paul
Meiji Seika Kaisha Ltd.
Zaidan Hojin Biseibutsu Kagaku Kenkyu Kai
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