9a, 11-3C-bicyclic 9a-azalide derivatives

Details 9a, 11-3C-bicyclic 9a-azalide derivatives 9a, 11-3C-bicyclic 9a-azalide derivatives

2007-10-02

2007-10-02

Peselev, Elli (Department: 1623)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Carbohydrate doai

C536S007400

Reexamination Certificate

active

10946339

ABSTRACT:
The present invention discloses compounds of formula I, or pharmaceutically acceptable salts, esters, or prodrugs thereof:which exhibit antibacterial properties. The present invention further relates to pharmaceutical compositions comprising the aforementioned compounds for administration to a subject in need of antibiotic treatment. The invention also relates to methods of treating a bacterial infection in a subject by administering a pharmaceutical composition comprising the compounds of the present invention. The invention further includes process by which to make the compounds of the present invention.

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Bright, G. Michael, et al., “Synthesis,In VitroandIn VivoActivity of Novel 9-Deoxo-9a-Aza-9a-Homoerythromycin A Derivatives; A New Class of Macrolide Antibiotics, the Azalides,”J. of Antibiotics, vol. XLI(8): 1029-1047 (1988).

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