Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...
Patent
1991-04-08
1993-11-02
Rizzo, Nicholas S.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Heterocyclic carbon compounds containing a hetero ring...
514202, 514206, 540221, 540222, 540225, 540226, 540227, C07D50157, A61K 31545
Patent
active
052583775
ABSTRACT:
Derivatives of 2-spirocyclopropyl 4-acylcephem sulfones of the formula (I) ##STR1## are provided which are useful as potent elastase inhibitors and hence are useful in the prevention, control and treatment of inflammatory conditions, especially arthritis and emphysema.
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Czajkowski David
Fiakpui Charles
Maiti Samarendra N.
Micetich Ronald G.
Reddy Narender A. V.
Rizzo Nicholas S.
Taiho Pharmaceutical Co. Ltd.
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