2,9-Dioxatricyclo[4,3,1,0.sup.3,7 ] decane derivatives, processe

Details 2,9-Dioxatricyclo[4,3,1,0.sup.3,7 ] decane derivatives, processe 2,9-Dioxatricyclo[4,3,1,0.sup.3,7 ] decane derivatives, processe

1978-04-19

1979-06-12

Love, Ethel G.

Drug, bio-affecting and body treating compositions

Nonspecific immunoeffector, per se ; or nonspecific...

2603403, A61K 31335

Patent

active

041580613

ABSTRACT:
3-Azidomethyl-2,9-dioxatricyclo[4,3,1,0.sup.3,7 ] decane derivatives are disclosed which exhibit analgesic, as well as antipyretic and antiphlogistic properties, and which have the formula (I) ##STR1## wherein: R.sub.1 represents alkyloxy or aralkyloxy;
One of R.sub.2 and R.sub.3 is hydrogen and the other represents hydroxy, acyloxy or carbamyloxy, or R.sub.2 and R.sub.3 jointly represent oxygen; and,
Y and y' each represent hydrogen or jointly form a bond,
As well as pharmaceutical formulations thereof.
By reducing the 3-azidomethyl compounds of formula (I), the corresponding 3-aminomethyl compounds are obtained which possess sedative properties and which are valuable intermediates for preparing 3-(mono- or dialkylaminomethyl)-2,9-dioxatricyclo[4,3,1,0.sup.3,7 ] decanes which exhibit sedative and soporific activities.

REFERENCES:
patent: 4016176 (1977-04-01), Thies
patent: 4089971 (1978-05-01), Thies

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