Bis-sulfonamide hydroxyethyl-amino retroviral protease...

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

Reexamination Certificate

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C514S233800, C514S234500, C514S253110, C514S249000, C514S252100, C514S317000, C514S321000, C514S394000, C544S160000, C544S383000, C544S360000, C544S367000, C544S368000, C544S370000, C549S065000, C549S438000, C549S366000, C549S467000, C546S270100, C546S234000, C546S198000, C546S293000, C564S078000, C564S082000

Reexamination Certificate

active

07091219

ABSTRACT:
Bis-sulfonamido hydroxyethylamino compounds are effective as retroviral protease inhibitors, and in particular as inhibitors of HIV protease. The present invention relates to retroviral protease inhibiting compounds of the formula:or a pharmaceutically acceptable salt, prodrug or ester thereof, wherein the variables are as defined herein.

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