Aromatase inhibitors from azoles

Details Aromatase inhibitors from azoles Aromatase inhibitors from azoles

1988-08-15

1989-07-04

Henderson, Christopher

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

548250, 548252, 548255, 548260, C07D 4106, C07D24904, C07D25704

Patent

active

048452270

ABSTRACT:
This invention provides azole derivatives, their pharmaceutical formulations, and their use in methods of inhibiting aromatase and treating or preventing estrogen-dependent diseases in mammals.

REFERENCES:
patent: 4094881 (1978-06-01), Berges
patent: 4098894 (1978-07-01), Buchal et al.
patent: 4227004 (1980-10-01), Wildonger
Chemical Abstracts 89:24368q (1978).
Chemical Abstracts 71:61296p.
Fisher, et al., "5-Aroyltetrazoles," J. Org. Chem., 24, 1650, (1959).
Burgess et al., "Synthesis . . . of . . . Azafulvenes," J. Org. Chem., 39(7), 940 (1974).
Adelstein, "Antiarrhythmic Agents . . . ", J. Med. Chem., 16(4), 309 (1973).
Balieu et al., "Tetrazole Analogues . . . ", Acta Chemica Scandinavica, 27, 1233 (1973); 26, 295 (1972).
Chemical Abstracts 89:179927v (1978).
Zaugg et al., "Reactions of Some Ester Alkaloids . . . ,"]J. Org. Chem., 23, 847 (1958).

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