Hexahydroindenopyridine compounds having antispermatogenic activ

Details Hexahydroindenopyridine compounds having antispermatogenic activ Hexahydroindenopyridine compounds having antispermatogenic activ

1993-08-16

1994-06-07

Ivy, C. Warren

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

546 79, C07D22116, A01N 4342, A61K 3144

Patent

active

053190840

ABSTRACT:
Hexahydroindenopyridine compounds having the following formula and relative stereochemistry ##STR1## where R.sup.1 is C.sub.1-6 alkyl, R.sup.2 is hydrogen or C.sub.1-6 alkyl and R.sup.3 is carboxyl or a group which is metabolized to a carboxyl group under mammalian physiological conditions exhibit potent antispermatogenic activity and are useful in a method of inhibiting spermatogenesis in mammals.

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