Novel cyclic Hexapeptide LHRH antagonists

Details Novel cyclic Hexapeptide LHRH antagonists Novel cyclic Hexapeptide LHRH antagonists

1985-02-08

1987-04-21

Phillips, Delbert R.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Peptide containing doai

514800, 530321, 530313, A61K 3743, C07K 512, C07K 720

Patent

active

046596917

ABSTRACT:
Novel peptides of the formula: ##STR1## where R.sup.1 through R.sup.8 are various radicals derived from L- and D- amino acids; having LHRH antagonist activity; useful in reducing fertility.
Pharmaceutical compositions and methods for use in reducing fertility.

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patent: 4377515 (1983-03-01), Veber et al.
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