Preparation of N-alkyl-N-pyridinyl-1H-indol-1-amines

Details Preparation of N-alkyl-N-pyridinyl-1H-indol-1-amines Preparation of N-alkyl-N-pyridinyl-1H-indol-1-amines

1995-05-31

1997-07-01

Fan, Jane

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

C07D40104

Patent

active

056440626

ABSTRACT:
The synthesis of memory enhancing, analgetic, and antidepressant N-alkyl-N-pyridinyl-1H-indol-1-amines is described.

REFERENCES:
patent: 4022795 (1977-05-01), Bamfield et al.
patent: 4389360 (1983-06-01), Sato et al.
patent: 4618686 (1986-10-01), Boyer
patent: 4692554 (1987-09-01), Yamaguchi et al.
patent: 4752610 (1988-06-01), Effland et al.
patent: 4880822 (1989-11-01), Effland et al.
patent: 4970218 (1990-11-01), Effland et al.
patent: 5032599 (1991-07-01), Effland et al.
patent: 5039811 (1991-08-01), Effland et al.
J.C. Powers, Journal of Organic Chemistry, 31, 2627 (1966), entitled "Chloroindoles" and published in the United States of America.
M. Somei and M. Natsume, Tetrahedron Letters, 461 (1974), entitled "1-Aminoindoles" and published in Great Britain.
M. R. Brennan, et al., Heterocycles, 24, 2879 (1986), entitled "The Preparation And Spectral Characterization of 2-Haloindoles, 3-Haloindoles, And 2,3-Dihaloindoles" and published in Japan.
M. Somei, et al., Chemical and Pharmaceutical Bulletin, 26, 2522 (1978), entitled "A Novel N-Amination Method and Its Application To the Preparation of N-aminoheterocycles" and published in Japan.
D. L. Comins and M. O. Killpack, Tetrahedron Letters, 30, 4337 (1989) entitled "N-methyl Lithiation of N-methylindoles Directed by .alpha.-Amino Alkoxides" and published in the United Kingdom.
G. M. Shutske. Medicinal Chemistry Approaches to Alzheimer's Disease and Other Dementias Symposium, Division of Educational Services, Mayo Clinic, Jacksonville, Jacksonville, Florida, Sep. 13, 1993.

Affiliated with

Also associated with

Rating

Preparation of N-alkyl-N-pyridinyl-1H-indol-1-amines does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Preparation of N-alkyl-N-pyridinyl-1H-indol-1-amines, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Preparation of N-alkyl-N-pyridinyl-1H-indol-1-amines will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFUS-PAI-O-598864