Antitumor antibiotics

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Peptide containing doai

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514 9, 514 2, 530317, A61K 3815, C07K 1102

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active

056438710

ABSTRACT:
The present invention relates to novel antitumor depsipeptides produced by Micromonospora strain 39500, ATCC 55011, and having the structural formula ##STR1## wherein R.sub.1 is 2-methylpropanoyl, and R.sub.2 is 2-methylppropanoyl, propanoyl or acetyl; or R.sub.1 is 3-methylbutanoyl, and R.sub.2 is 2-methylpropanoyl or 3-methylbutanoyl; or R.sub.1 is propanoyl, and R.sub.2 is acetyl or propanoyl.

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