11β-hydroxysteroid dehydrogenase type 1 active compounds

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

Reexamination Certificate

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C514S317000, C546S184000, C546S192000

Reexamination Certificate

active

08053447

ABSTRACT:
A novel class of compounds of the general formula (I), their use in therapy, pharmaceutical compositions comprising the compounds, as well as their use in the manufacture of medicaments are described. The present compounds modulate the activity of 11β-hydroxy-steroid dehydrogenase type 1 (11βHSD1) and are accordingly useful in the treatment of diseases in which such a modulation is beneficial, e.g. the metabolic syndrome.

REFERENCES:
patent: 2913454 (1959-11-01), Petersen et al.
patent: 3723442 (1973-03-01), Nakanishi et al.
patent: 3784551 (1974-01-01), Nakanishi et al.
patent: 4350696 (1982-09-01), Cross et al.
patent: 4482555 (1984-11-01), Doria et al.
patent: 4851423 (1989-07-01), Girijavallabhan et al.
patent: 4963590 (1990-10-01), Backstrom et al.
patent: 5001133 (1991-03-01), Richardson et al.
patent: 5049695 (1991-09-01), Abraham et al.
patent: 5112861 (1992-05-01), Backstrom et al.
patent: 5122539 (1992-06-01), Abraham et al.
patent: 5169850 (1992-12-01), Dusza et al.
patent: 5225402 (1993-07-01), Ogawa et al.
patent: 5258407 (1993-11-01), Washburn et al.
patent: 5260325 (1993-11-01), Markwalder et al.
patent: 5272167 (1993-12-01), Girijavallabhan et al.
patent: 5274104 (1993-12-01), Arnaud et al.
patent: 5290803 (1994-03-01), Abraham et al.
patent: 5314880 (1994-05-01), Whittaker et al.
patent: 5356904 (1994-10-01), Freidinger et al.
patent: 5382680 (1995-01-01), Abraham et al.
patent: 5426105 (1995-06-01), Manning et al.
patent: 5432191 (1995-07-01), Abraham et al.
patent: 5436254 (1995-07-01), Ogawa et al.
patent: 5446194 (1995-08-01), Backstrom et al.
patent: 5459144 (1995-10-01), Girijavallabhan et al.
patent: 5585394 (1996-12-01), Di Malta et al.
patent: 5591892 (1997-01-01), Abraham et al.
patent: 5596020 (1997-01-01), Morris et al.
patent: 5602137 (1997-02-01), Ruhter et al.
patent: 5648375 (1997-07-01), Abraham et al.
patent: 5650513 (1997-07-01), Langhals et al.
patent: 5652247 (1997-07-01), Ogawa et al.
patent: 5674879 (1997-10-01), Manning et al.
patent: 5677330 (1997-10-01), Abraham et al.
patent: 5705521 (1998-01-01), Abraham et al.
patent: 5731454 (1998-03-01), Abraham et al.
patent: 5750532 (1998-05-01), Girijavallabhan et al.
patent: 5786379 (1998-07-01), Bernardon
patent: 5795907 (1998-08-01), Kalindjian et al.
patent: 5872282 (1999-02-01), Abraham et al.
patent: 5912260 (1999-06-01), Kalindjian et al.
patent: 5919829 (1999-07-01), Kalindjian et al.
patent: 5927283 (1999-07-01), Abraham et al.
patent: 5932569 (1999-08-01), Janssens et al.
patent: 5939437 (1999-08-01), Kalindjian et al.
patent: 6001879 (1999-12-01), Seitz et al.
patent: 6096736 (2000-08-01), Ogawa et al.
patent: 6124289 (2000-09-01), He et al.
patent: 6458803 (2002-10-01), Sikorski et al.
patent: 6506783 (2003-01-01), Camden
patent: 6521641 (2003-02-01), Klein et al.
patent: 6548549 (2003-04-01), Seitz et al.
patent: 6613803 (2003-09-01), Wang et al.
patent: 6638947 (2003-10-01), Wang et al.
patent: 6696442 (2004-02-01), Wang et al.
patent: 6833371 (2004-12-01), Atkinson et al.
patent: 7129242 (2006-10-01), Satoh et al.
patent: 7157490 (2007-01-01), Colandrea et al.
patent: 7186735 (2007-03-01), Strobel et al.
patent: 7265122 (2007-09-01), Wu et al.
patent: 7358238 (2008-04-01), Andersen et al.
patent: 7501405 (2009-03-01), Kampen et al.
patent: 7557110 (2009-07-01), Kataoka et al.
patent: 7700583 (2010-04-01), Gundertofte et al.
patent: 7723323 (2010-05-01), Andersen et al.
patent: 2002/0006932 (2002-01-01), Galley et al.
patent: 2002/0115671 (2002-08-01), Goehring
patent: 2003/0144256 (2003-07-01), Klein et al.
patent: 2004/0142922 (2004-07-01), Alanine et al.
patent: 2004/0186102 (2004-09-01), Wu et al.
patent: 2005/0009871 (2005-01-01), Ramesh et al.
patent: 2005/0054850 (2005-03-01), Wu et al.
patent: 2005/0080087 (2005-04-01), Pendri et al.
patent: 2005/0154202 (2005-07-01), Hagmann et al.
patent: 2005/0261302 (2005-11-01), Hoff et al.
patent: 2006/0009918 (2006-01-01), Mallik et al.
patent: 2006/0079506 (2006-04-01), Linders et al.
patent: 2006/0094699 (2006-05-01), Kampen et al.
patent: 2006/0111366 (2006-05-01), Andersen et al.
patent: 2006/0149070 (2006-07-01), Rohde et al.
patent: 2006/0281773 (2006-12-01), Patel et al.
patent: 2007/0054882 (2007-03-01), Klein et al.
patent: 2007/0270408 (2007-11-01), Andersen et al.
patent: 2008/0108598 (2008-05-01), Andersen et al.
patent: 2009/0105289 (2009-04-01), Kilburn et al.
patent: 2009/0118259 (2009-05-01), Kilburn et al.
patent: 2009/0124598 (2009-05-01), Andersen et al.
patent: 2009/0137574 (2009-05-01), Kampen et al.
patent: 2009/0264412 (2009-10-01), Kampen et al.
patent: 2009/0264414 (2009-10-01), Andersen et al.
patent: 2009/0306048 (2009-12-01), Kilburn et al.
patent: 2009/0325932 (2009-12-01), Ebdrup et al.
patent: 2010/0056600 (2010-03-01), Ebdrup et al.
patent: 2010/0076041 (2010-03-01), Kilburn et al.
patent: 2010/0087543 (2010-04-01), Ebdrup et al.
patent: 2010/0120743 (2010-05-01), Gundertofte et al.
patent: 2010/0137377 (2010-06-01), Petersen et al.
patent: 2010/0168083 (2010-07-01), Ebdrup
patent: 2010/0197658 (2010-08-01), Andersen et al.
patent: 2010/0331366 (2010-12-01), Ebdrup
patent: 2011/0003852 (2011-01-01), Ebdrup
patent: 2011/0003856 (2011-01-01), Ebdrup
patent: 2011/0039853 (2011-02-01), Ebdrup
patent: 1736485 (2006-02-01), None
patent: 4338784 (1995-05-01), None
patent: 1 669 350 (2006-06-01), None
patent: 2456731 (1980-12-01), None
patent: 825514 (1956-11-01), None
patent: 08-048662 (1996-02-01), None
patent: 09-221476 (1997-08-01), None
patent: 11-152269 (1999-06-01), None
patent: 2001 139574 (2001-05-01), None
patent: 2003-286171 (2003-10-01), None
patent: 2007-231005 (2007-09-01), None
patent: WO 94/01113 (1994-01-01), None
patent: WO 94/18193 (1994-08-01), None
patent: WO 97/07789 (1997-03-01), None
patent: WO 97/22588 (1997-06-01), None
patent: WO 97/24328 (1997-07-01), None
patent: WO 98/46559 (1998-10-01), None
patent: WO 99/30699 (1999-06-01), None
patent: WO 99/61013 (1999-12-01), None
patent: WO 00/12074 (2000-03-01), None
patent: WO 00/46197 (2000-08-01), None
patent: WO 00/47558 (2000-08-01), None
patent: WO 00/63165 (2000-10-01), None
patent: WO 00/73283 (2000-12-01), None
patent: WO 01/02385 (2001-01-01), None
patent: WO 01/22969 (2001-04-01), None
patent: WO 01/32621 (2001-05-01), None
patent: WO 01/44213 (2001-06-01), None
patent: WO 01/64676 (2001-09-01), None
patent: WO 01/90090 (2001-11-01), None
patent: WO 01/90091 (2001-11-01), None
patent: WO 01/90092 (2001-11-01), None
patent: WO 01/90093 (2001-11-01), None
patent: WO 01/90094 (2001-11-01), None
patent: WO 02/00626 (2002-01-01), None
patent: WO 02/02797 (2002-01-01), None
patent: WO 02/10191 (2002-02-01), None
patent: WO 02/072084 (2002-09-01), None
patent: WO 02/076435 (2002-10-01), None
patent: WO 02/094799 (2002-11-01), None
patent: WO 20/089781 (2002-11-01), None
patent: WO 02/100819 (2002-12-01), None
patent: WO 03/000649 (2003-01-01), None
patent: WO 03/028641 (2003-04-01), None
patent: WO 03/028730 (2003-04-01), None
patent: WO 03/029246 (2003-05-01), None
patent: WO 03/037274 (2003-05-01), None
patent: WO 03/037900 (2003-05-01), None
patent: WO 03/065983 (2003-08-01), None
patent: WO 03/070732 (2003-08-01), None
patent: WO 03/086410 (2003-10-01), None
patent: WO 2004/024896 (2004-03-01), None
patent: WO 2004/024897 (2004-03-01), None
patent: WO 2004/033427 (2004-04-01), None
patent: WO 2004/052461 (2004-06-01), None
patent: WO 2004/056744 (2004-07-01), None
patent: WO 2004/056745 (2004-07-01), None
patent: WO 2004/065351 (2004-08-01), None
patent: WO 2004/075823 (2004-09-01), None
patent: WO 2004/087159 (2004-10-01), None
patent: WO 2004/089380 (2004-10-01), None
patent: WO 2004/089415 (2004-10-01), None
patent: WO 2004/089416 (2004-10-01), None
patent: WO 2004/089470 (2004-10-01), None
patent: WO 2004/089471 (2004-10-01), None
patent: WO 2004/089896 (2004-10-01), None
patent: WO2004/089896 (2004-10-01), None
patent: WO 2004/091610 (2004-10-01), None
patent: WO 2005/013950 (2005-02-01), None
patent: WO 2005/032484 (2005-04-01), None
patent: WO 2005/035534 (2005-04-01), None
patent: WO 2005/085202 (2005-09-01),

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