Gyrase inhibitors and uses thereof

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...

Reexamination Certificate

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C514S234500, C514S252140, C514S252190, C514S256000, C514S269000, C514S275000, C514S293000, C514S303000, C514S314000, C514S318000, C514S322000, C514S338000, C514S364000, C514S375000, C514S395000, C540S578000, C544S122000, C544S124000, C544S324000, C544S330000, C544S331000, C544S333000, C546S082000, C546S118000, C546S167000, C546S193000, C546S199000, C546S271700, C546S273100, C546S273400, C548S143000, C548S222000, C548S304700, C548S305100, C548S308100

Reexamination Certificate

active

07414046

ABSTRACT:
The present invention relates to compounds of the formula I:or a pharmaceutically acceptable derivative or prodrug thereof. The compounds are useful as inhibitors of bacterial gyrase activity. The present invention also relates to methods for treating bacterial infections in mammala. The present invention also relates to methods for decreasing bacterial quantity in a biological sample.

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