Organic compounds -- part of the class 532-570 series – Organic compounds – Carbohydrates or derivatives
Reexamination Certificate
2007-11-20
2007-11-20
Jiang, S. Anna (Department: 1623)
Organic compounds -- part of the class 532-570 series
Organic compounds
Carbohydrates or derivatives
C536S027300, C536S124000
Reexamination Certificate
active
10471682
ABSTRACT:
An improved process for preparing N6 -substituted aminopurine ribofuranose nucleosides. Compounds of this type are known to be usefull in the prepartation of compounds having activitity at adenosine receptors, e.g. Adenosine A1 receptor. The process comprises the step of reacting a 6-halopurine ribofuranose nucleoside with an amine in the presence of CaCO3 , wherein acid is added to the reaction mixture.
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Berry Malcolm
Roberts John C.
Xie Shiping
Crane L. E.
Deppenbrock Bonnie L.
Glaxo Group Limited
Jiang S. Anna
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