Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...
Reexamination Certificate
2007-03-13
2007-03-13
Dentz, Bernard (Department: 1625)
Organic compounds -- part of the class 532-570 series
Organic compounds
Heterocyclic carbon compounds containing a hetero ring...
C564S373000
Reexamination Certificate
active
10962746
ABSTRACT:
A synthesis is described for intermediates which are readily amenable to the large scale preparation of hydroxyethylurea-based chiral HIV protease inhibitors. The method includes forming a diastereoselective epoxide from a chiral alpha amino aldehyde.
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Getman Daniel P.
Mueller Richard A.
Ng John S.
Przybyla Claire A.
Vazquez Michael L.
Banner & Witcoff Ltd
Dentz Bernard
G.D. Searle & Co.
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