Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Reexamination Certificate
2006-12-05
2006-12-05
Aulakh, Charanjit S. (Department: 1625)
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
C546S143000, C546S146000, C546S139000, C514S307000
Reexamination Certificate
active
07144895
ABSTRACT:
Compounds having the formula (I),and pharmaceutically-acceptable salts, hydrates, or prodrugs thereof, are useful as serine protease inhibitors, wherein X is —OH, —O(alkyl), —O(aryl), —O(arylalkyl), —NR5(aryl), or —NR5(arylalkyl); W is hydrogen or —(CR7R8)q—W1; W1is hydrogen or a bond with R6; Z is a 5-membered heteroaryl group, a five to six membered heterocyclo or cycloalkyl group, a 9 to 10 membered bicyclic aryl or heteroaryl, or a six membered aryl or heteroaryl, and R1, R2, R3, R5, R6, R7, and R16are as defined in the specification.
REFERENCES:
patent: 6140353 (2000-10-01), Ackermann et al.
patent: 6194409 (2001-02-01), Van Boeckel et al.
patent: 6242644 (2001-06-01), Ackermann et al.
patent: 6335324 (2002-01-01), Bisacchi et al.
patent: 6358960 (2002-03-01), Senokuchi et al.
patent: 6472393 (2002-10-01), Aliagas-Martin et al.
patent: 6642252 (2003-11-01), Bisacchi et al.
patent: 6699994 (2004-03-01), Babu et al.
patent: WO 96/20689 (1996-07-01), None
patent: WO 97/10214 (1997-03-01), None
patent: WO 01/44172 (2001-06-01), None
patent: WO 01/90051 (2001-11-01), None
patent: WO 02/09688 (2002-02-01), None
patent: WO 2002/034711 (2002-05-01), None
patent: WO2003013531 (2003-02-01), None
patent: WO 03/66588 (2003-08-01), None
patent: WO 2003/084533 (2003-10-01), None
patent: WO 2004/072101 (2004-08-01), None
U.S. Appl. No. 10/775,923, filed Feb. 10, 2004, Glunz et al.
Stedman's Medical Dictionary, 27thEdition Illustrated in Color, Lippincott Williams & Wilkins, 1999, pp. 1711, 1831, 1832.
Dorland's Illustrated Medical Dictionary, 29thEdition, W.B. Saunders Company, 2000, pp. 1836, 1837.
Robbins Pathologic Basis of Disease, Sixth Edition, W. B. Saunders Company, 1999, pp. 113-138.
Hurst's The Heart, 10thEdition, 2001, pp. 1373-1384.
Harrison's Principles of Internal Medicine, 14thEdition, vol. 2, 1998, pp. 2325-2348.
Bisacchi Gregory S.
Morton George C.
Aulakh Charanjit S.
Bristol-Myers Squibb Co.
Sun Jing G.
Winstow Anastasia P.
LandOfFree
Benzene acetamide compounds useful as serine protease... does not yet have a rating. At this time, there are no reviews or comments for this patent.
If you have personal experience with Benzene acetamide compounds useful as serine protease..., we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Benzene acetamide compounds useful as serine protease... will most certainly appreciate the feedback.
Profile ID: LFUS-PAI-O-3718896