Method for the preparation of citalopram

Details Method for the preparation of citalopram Method for the preparation of citalopram

2006-04-18

2006-04-18

Dentz, Bernard (Department: 1625)

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

Reexamination Certificate

active

07030252

ABSTRACT:
A method for the preparation of citalopram comprising reductive hydrolysis of a compound of Formula (IV)wherein R is a N,N-disubstituted amid group or an optionally substituted 4,5-dihydro-1,3-oxazol-2-yl group, and conversion of the resulting 5-formyl compound to citalopram.

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