Method for preparing intermediates useful in synthesis of...

Details Method for preparing intermediates useful in synthesis of... Method for preparing intermediates useful in synthesis of...

2005-12-13

2005-12-13

Dentz, Bernard (Department: 1625)

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

C548S465000, C548S517000, C549S215000

Reexamination Certificate

active

06974876

ABSTRACT:
A synthesis is described for intermediates which are readily amenable to the large scale preparation of hydroxyethylurea-based chiral HIV protease inhibitors. The method includes forming a diastereoselective epoxide from a chiral alpha amino aldehyde.

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