Dermorphin analogs having pharmacological activity

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Peptide containing doai

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530330, A61K 3800, A61K 3802, C07K 500, C07K 700

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active

056021003

ABSTRACT:
This invention relates to novel dermorphin analogs having pharmacological activity. More particularly, this invention relates to novel tetrapeptides having specific structural features and a net charge of +2 or greater. The peptides of this invention are useful in treating pain and gastro-intestinal disorders. Accordingly, this invention also relates to pharmaceutical compositions comprising those peptides and methods for treating pain and gastro-intestinal disorders.

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