Methods of modulating pharmacokinetics of oligonucleotides

Organic compounds -- part of the class 532-570 series – Organic compounds – Carbohydrates or derivatives

Reexamination Certificate

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C536S024300, C536S025300

Reexamination Certificate

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06921812

ABSTRACT:
2′-O-(2-Methylthioethyl), has been incorporated into oligonucleotides and evaluated for antisense properties in comparison with the known 2′-O-(2-methoxyethyl) 2′-O-MOE modification. The 2′-O-MTE modified oligonucleotides exhibit improved binding to human serum albumin compared with the 2′-O-MOE modified oligonucleotides and maintain high binding affinity to target RNA.

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