Organic compounds -- part of the class 532-570 series – Organic compounds – Nitrogen attached directly or indirectly to the purine ring...
Reexamination Certificate
2011-08-02
2011-08-02
Wilson, James O (Department: 1624)
Organic compounds -- part of the class 532-570 series
Organic compounds
Nitrogen attached directly or indirectly to the purine ring...
Reexamination Certificate
active
07989623
ABSTRACT:
The compound of formula (8), in racemic or single enantiomeric form, is useful in making N-(diphenylmethyl)-piperazines such as cetirizine and levocetrizine.wherein Z is preferably phenyl.
REFERENCES:
patent: 4525358 (1985-06-01), Baltes et al.
patent: 5478941 (1995-12-01), Cossement et al.
patent: 5698558 (1997-12-01), Gray
patent: 1139113 (1962-11-01), None
patent: 617028 (1994-09-01), None
patent: 955295 (1999-11-01), None
patent: 1 236 722 (2002-09-01), None
patent: 2 076 403 (1981-12-01), None
patent: 2 225 321 (1990-05-01), None
patent: WO 94/06429 (1994-03-01), None
patent: WO 2007/066163 (2007-06-01), None
M. Gillard et al., “Binding Characteristics of Cetirizine and Levocetirizine to Human H1 Histamine Receptors: Contribution of Lys191 and Thr194”, Molecular Pharmacology 61:391-399, 2002.
G. R. Clemo et al., “The Optical Rotary Powers of Some 4-Substituted Benzhydrylamines” J. Chem. Soc. 1939 pp. 1958-1960.
C. J. Opalka “A Novel Synthesis of the Enantiomers of an Antihistamine Drug by Piperazine Formation from a Primary Amine”, Synthesis, Jul. 1995 (7) pp. 766-768.
A. P. Sineokov, et al., Ref.zh.Khim., 1971, Abstr. No. 6Zh476 (Chem. Abstract XP-002464434).
P. Bercot, Compt. Rend. (1964), 258(1), 224-6 (Chem. Abstract XP-002464436).
N. Suciu, Revue Roumaine de Chimie (1966) 11(6), 745-9 (Chem. Abstract XP-002464437).
G. Olah, Acta Chimica Acad. Sci. Hung. (1955), 7, 443-9 (Chem. Abstract XP-002464438).
K. Yoon, Bioorganic and Medicinial Chemistry (2003), 11(15), 3237-3244 (Chem. Abstract XP-002464439).
Chemical Abstracts XP-002464435 (Mar. 28, 2003).
Leeser Erich A
Muncy Geissler Olds & Lowe, PLLC
Synthon BV
Wilson James O
LandOfFree
Process for making n-(diphenylmethyl)piperazines does not yet have a rating. At this time, there are no reviews or comments for this patent.
If you have personal experience with Process for making n-(diphenylmethyl)piperazines, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Process for making n-(diphenylmethyl)piperazines will most certainly appreciate the feedback.
Profile ID: LFUS-PAI-O-2796205