Chemistry: natural resins or derivatives; peptides or proteins; – Proteins – i.e. – more than 100 amino acid residues – Plant proteins – e.g. – derived from legumes – algae or...
Reexamination Certificate
2011-08-30
2011-08-30
Steele, Amber D. (Department: 1639)
Chemistry: natural resins or derivatives; peptides or proteins;
Proteins, i.e., more than 100 amino acid residues
Plant proteins, e.g., derived from legumes, algae or...
C530S321000, C530S323000, C530S331000, C530S332000, C514S018700, C930S010000, C930S020000, C930S080000, C930S270000
Reexamination Certificate
active
08008440
ABSTRACT:
A library of macrocyclic compounds of the formula (I)where part (A) is a bivalent radical, a —(CH2)y— bivalent radical or a covalent bond;where part (B) is a bivalent radical, a —(CH2)z— bivalent radical, or a covalent bond;where part (C) is a bivalent radical, a —(CH2)t— bivalent radical, or a covalent bond; andwhere part (T) is a —Y-L-Z- radical wherein Y is CH2or CO, Z is NH or O and L is a bivalent radical. These compounds are useful for carrying out screening assays or as intermediates for the synthesis of other compounds of pharmaceutical interest. A process for the preparation of these compounds in a combinatorial manner, is also disclosed.
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Berthiaume Gilles
Deslongchamps Pierre
Dory Yves
Lan Ruoxi
Ouellet Luc
Myers Bigel & Sibley Sajovec, PA
Steele Amber D.
Tranzyme Pharma Inc.
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