Phenylpyridone derivative

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

Reexamination Certificate

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Details

C514S235500, C514S318000, C514S333000, C514S343000, C546S300000, C546S261000, C546S194000, C546S276400, C546S256000, C544S131000

Reexamination Certificate

active

07875633

ABSTRACT:
A compound represented by the formula (I) is contained as an active ingredient:wherein R1and R2independently represent a hydrogen atom, a lower alkyl group or the like, or R1together with a nitrogen atom to which L, Z2and R1are attached may form an aliphatic nitrogenated heterocyclic group and R1and R2together with a nitrogen atom to which they are attached may form an aliphatic nitrogenated heterocyclic group; X represents a methine group or a nitrogen atom; Y represents —CH2—O—, —CH═CH— or the like; Z1represents a single bond, a C1-4alkylene group or the like; Z2represents a single bond or a C1-4alkylene group; L represents a methylene group, a C3-8cycloalkylene group or the like; and Ar represents an aromatic carbocyclic group or the like. The compound is useful as a pharmaceutical for a central nerves system disease, a cardiovascular disease or a metabolic disease.

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