Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...
Patent
1993-10-08
1995-07-18
Rizzo, Nicholas
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Heterocyclic carbon compounds containing a hetero ring...
540205, 540310, 540222, C07D47104, A61K 31435
Patent
active
054341477
ABSTRACT:
Antimicrobial quinolonyl lactam esters comprising a lactam-containing moiety linked, by an ester group, to the 3-carboxy group of a quinolone moiety. These compounds are of the formula: ##STR1## wherein (1) R.sup.3, R.sup.4, and R.sup.5, together with bonds "a" and "b", form certain lactam-containing moieties similar to those known in the art to have antimicrobial activity; and
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Demuth, Jr. Thomas P.
White Ronald W.
Clark Karen F.
Proctor & Gamble Pharmaceuticals, Inc.
Rizzo Nicholas
Suter David L.
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