3-alkyloxy-, aryloxy-, or arylalkyloxy-benzo [.beta.]thiophene-2

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

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549 52, 549 53, 549 54, 549 55, A61K 3138, C07D33368

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active

053569261

ABSTRACT:
3-Alkyloxy-, aryloxy-, or arylalkyloxybenzo[b]-thiophene-2-carboxamides are described as agents which block leukocyte adherence to vascular endothelium and, as such, are effective therapeutic agents for treating inflammatory diseases. Certain of these compounds are novel and methods of preparation are also described.

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