Polycyclic fused ring modulators of acetylcholine receptors

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

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514293, 546 81, 546 83, 546 84, 546 88, A61K 3144, C07D47104, C07D491147

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active

055677100

ABSTRACT:
In accordance with the present invention, there is provided a class of polycyclic fused ring compounds which are modulators of acetylcholine receptors. The compounds of the invention displace acetylcholine receptor ligands from their binding sites. Invention compounds may act as agonists, partial agonists, antagonists or allosteric modulators of acetylcholine receptors.

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