Pyrazolo[1,5-a]-1,3,5-triazines

Details Pyrazolo[1,5-a]-1,3,5-triazines Pyrazolo[1,5-a]-1,3,5-triazines

Filed on

1984-05-25

Date issued

1986-01-21

Examiner

Ford, John M.

Patent Class

Drug, bio-affecting and body treating compositions

SubClass

Designated organic active ingredient containing

SubSubClass

Heterocyclic carbon compounds containing a hetero ring...

Other Related Categories

544211, 544212, 544113, 544206, 544245, 544197, 544198, 544207, 544219, 544216, 544180, C07D48704, C07D40314, C07D40714, A61K 31415

Type

Patent

Status

active

Patent number

045658153

Description

ABSTRACT:
A compound having anti-ulcer activity and having the formula ##STR1## wherein D is H, SH, NH.sub.2, OH, R.sup.4 S where R.sup.4 is a lower alkyl group; E is OH or NH.sub.2 ; J is H or aryl; X is CH or N; Y is CH, N, or CT, wherein T is a halogen; Z is CH or N; A is ##STR2## and replaces a hydrogen of D, X, or E; R.sup.1 is H or CH.sub.3 ; L is CH.sub.2 S; Q is O or CH.sub.2 S; n is 0 or 1; 2 m 4; each R.sup.2 and R.sup.3, independently, is H, lower alkyl, cycloalkyl, or arylalkyl; or R.sup.2 and R.sup.3, together with the nitrogen atom to which they are attached, form a 4, 5, or 6 membered heterocyclic ring containing 0, 1, or 2 oxygen atoms and 1, 2, or 3 nitrogen atoms and being unsubstituted or lower alkyl substituted; or a pharmaceutically acceptable salt thereof.

REFERENCES:
patent: 4128658 (1978-12-01), Price et al.
Lumma et al. (1982) J. Med. Chem., 25 207-210.
Algieri et al. (1982) J. Med. Chem. 25 210-212.

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