Mercapto-imidazolyl derivatives

Details Mercapto-imidazolyl derivatives Mercapto-imidazolyl derivatives

1998-11-17

2000-09-05

Higel, Floyd D.

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

514341, 514383, 514397, 514399, 514400, 5462744, 2482686, 2483111, 2483154, 2483157, 2483251, 2483295, C07D23384, A01N 4350

Patent

active

061145394

DESCRIPTION:

BRIEF SUMMARY
TECHNICAL FIELD OF THE INVENTION

The present invention relates to new mercapto-imidazolyl derivatives, to a plurality of processes for their preparation, and to their use as microbicides.


BACKGROUND OF THE INVENTION

It has already been disclosed that a large number-of imidazolyl derivatives have fungicidal properties (cf. EP-A 0 015 756, EP-A 0 040 345, EP-A 0 052 424, EP-A 0 061 835, EP-A 0 297 345, EP-A 0 094 564, EP-A 0 196 038, EP-A 0 267 778, EP-A 0 378 953, EP-A 0 044 605, EP-A 0 069 442, EP-A 0 055 833, EP-A 0 301 393, DE-A 2 324 010, DE-A 2 737 489, DE-A 2 551 560, EP-A 0 065 485, DE-A 2 735 872, EP-A 0 234 242, DE-A 2 201 063, EP-A 0 145 294 and DE-A 3 721 786). While the activity of these substances is good, it leaves something to be desired in some cases at low rates of application.


DETAILED DESCRIPTION OF THE INVENTION

There have now been found new mercapto-imidazolyl derivatives of the formula ##STR1## in which R represents hydrogen or alkyl having 1 to 4 carbon atoms and ##STR2##
where substituted alkyl, optionally substituted alkenyl, optionally substituted cycloalkyl, optionally substituted aralkyl, optionally substituted aralkenyl, optionally substituted aroxyalkyl, optionally substituted aryl or optionally substituted heteroaryl,
or ##STR3##
where to 4 carbon atoms and 1 to 5 halogen atoms, cycloalkyl having 3 to 7 carbon atoms which is optionally substituted by halogen, or represents naphthyl, or represents phenyl which is optionally monosubstituted to trisubstituted by identical or different substituents from the series consisting of halogen, nitro, phenyl, phenoxy, alkyl having 1 to 4 carbon atoms, alkoxy having 1 to 4 carbon atoms, halogenoalkyl having 1 to 4 carbon atoms and 1 to 5 halogen atoms, halogenoalkoxy having 1 to 4 carbon atoms and 1 to 5 halogen atoms and/or halogenoalkylthio having 1 to 4 carbon atoms and 1 to 5 halogen atoms, and trisubstituted by identical or different substituents from the series consisting of halogen, alkyl having 1 to 4 carbon atoms, alkoxy having 1 to 4 carbon atoms, halogenoalkyl having 1 to 4 carbon atoms and 1 to 5 halogen atoms, halogenoalkoxy having 1 to 4 carbon atoms and 1 to 5 halogen atoms and/or halogenoalkylthio having 1 to 4 carbon atoms and 1 to 5 halogen atoms,
or ##STR4##
where alkyl having 1 to 6 carbon atoms, 1 to 4 carbon atoms, phenyl, phenoxy, halogenoalkyl having 1 to 4 carbon atoms and 1 to 5 halogen atoms, halogenoalkoxy having 1 to 4 carbon atoms and 1 to 5 halogen atoms, or represents halogenoalkylthio having 1 to 4 carbon atoms and 1 to 5 halogen atoms, and
or ##STR5##
where alkyl having 1 to 6 carbon atoms, alkoxy having 1 to 4 carbon atoms, halogenoalkyl having 1 to 4 carbon atoms and 1 to 5 halogen atoms, halogenoalkoxy having 1 to 4 carbon atoms and 1 to halogen atoms, or phenyl,
or ##STR6##
where 1 to 6 carbon atoms and 1 to 5 halogen atoms, cycloalkyl having 3 to 6 carbon atoms which is optionally substituted by halogen and/or alkyl having 1 to 4 carbon atoms, or represents optionally substituted aryl, or represents optionally substituted aralkyl,
or ##STR7##
where 1 to 4 carbon atoms, alkylthio having 1 to 4 carbon atoms, halogenoalkyl having 1 to 4 carbon atoms and 1 to 5 halogen atoms, halogenoalkoxy having 1 to 4 carbon atoms and 1 to 5 halogen atoms, halogenoalkylthio having 1 to 4 carbon atoms and 1 to 5 halogen atoms, phenyl which is optionally substituted by halogen and/or alkyl having 1 to 4 carbon atoms, or represents phenoxy which is optionally substituted by halogen and/or alkyl having 1 to 4 carbon atoms,
or ##STR8##
where 1 to 4 carbon atoms and 1 to 5 halogen atoms, cycloalkyl having 3 to 7 carbon atoms which is optionally substituted by halogen and/or alkyl having 1 to 4 carbon atoms, or represents cycloalkylalkyl having 3 to 7 carbon atoms in the cycloalkyl moiety and 1 to 4 carbon atoms in the alkyl moiety, or represents phenyl which is optionally substituted by halogen, or represents benzyl which is optionally substituted by halogen, having 1 to 4 carbon atoms, alkylthio having 1 to 4 carbon

REFERENCES:
patent: 3912752 (1975-10-01), Meiser et al.
patent: 3952002 (1976-04-01), Kramer et al.
patent: 4048318 (1977-09-01), Meiser et al.
patent: 4079062 (1978-03-01), Van Reet et al.
patent: 4147791 (1979-04-01), Meiser et al.
patent: 4205075 (1980-05-01), Baldwin et al.
patent: 4243405 (1981-01-01), Balasubramanyan et al.
patent: 4464381 (1984-08-01), Janssen et al.
patent: 4532341 (1985-07-01), Holmwood et al.
patent: 4549900 (1985-10-01), Kramer et al.
patent: 4598085 (1986-07-01), Heeres et al.
patent: 4626595 (1986-12-01), Holmwood et al.
patent: 4652580 (1987-03-01), Janssen et al.
patent: 4723984 (1988-02-01), Holmwood et al.
patent: 4789672 (1988-12-01), Holmwood et al.
patent: 4871390 (1989-10-01), Holmwood et al.
patent: 4897107 (1990-01-01), Holmwood et al.
patent: 4904297 (1990-02-01), Holmwood et al.
patent: 4906652 (1990-03-01), Karbach et al.
patent: 4911746 (1990-03-01), Holmwood et al.
patent: 4913727 (1990-04-01), Stroech et al.
patent: 4952232 (1990-08-01), Cuomo et al.
patent: 4965280 (1990-10-01), Cuomo et al.
patent: 4965281 (1990-10-01), Cuomo et al.
patent: 4968712 (1990-11-01), Elbe et al.
patent: 4980488 (1990-12-01), Stroech et al.
patent: 4988819 (1991-01-01), Stroech et al.
patent: 4990677 (1991-02-01), Stroech et al.
patent: 5034052 (1991-07-01), Stroech et al.
patent: 5081141 (1992-01-01), Colle et al.
patent: 5084465 (1992-01-01), Cuomo et al.
patent: 5087635 (1992-02-01), Shaber
patent: 5097047 (1992-03-01), Stroech et al.
patent: 5256683 (1993-10-01), Hutt et al.
patent: 5266585 (1993-11-01), Hubele et al.
patent: 5380743 (1995-01-01), Hutt et al.
patent: 5639918 (1997-06-01), Hutt et al.
patent: 5789430 (1998-08-01), Jautlat et al.
Chemical Abstracts, vol. 89, No. 13, Sep. 25, 1978, Abstract No. 109238 M.V. Postyanoi et al.

Affiliated with

Also associated with

Rating

Mercapto-imidazolyl derivatives does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Mercapto-imidazolyl derivatives, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Mercapto-imidazolyl derivatives will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFUS-PAI-O-2213568