Substituted 1,5-cyclohexadiene carboxylic acid derivatives

Details Substituted 1,5-cyclohexadiene carboxylic acid derivatives Substituted 1,5-cyclohexadiene carboxylic acid derivatives

1978-01-12

1980-02-05

Thomas, Jr., James O.

Drug, bio-affecting and body treating compositions

Antigen, epitope, or other immunospecific immunoeffector

Recombinant or stably-transformed bacterium encoding one or...

26050111, 424309, 424316, 424319, 424300, 424320, 424324, 560 47, 560 48, 560115, 560125, 562456, 562457, 562510, A61K 31215, C07C 6122

Patent

active

041873165

ABSTRACT:
Compounds of the following general formula and salts thereof are irreversible inhibitors of .gamma.-aminobutyric acid transaminase: ##STR1## wherein R.sub.1 is hydrogen, alkylcarbonyl wherein the alkyl moiety has from 1 to 4 carbon atoms and is straight or branched, alkoxycarbonyl wherein the alkoxy moiety has from 1 to 4 carbon atoms and is straight or branched, the radical ##STR2## wherein R.sub.4 is hydrogen, a straight or branched alkyl group having from 1 to 4 carbon atoms, benzyl or p-hydroxybenzyl; R.sub.2 is hydroxy, a straight or branched alkoxy group of from 1 to 8 carbon atoms, the group

REFERENCES:
patent: 3959356 (1976-05-01), Metcalf
patent: 3960927 (1976-06-01), Metcalf
Rando and Bangerter, J.A.C.S., 98, 6762 (1976).

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