Tricyclic compounds as TXA.sub.2 antagonists

Details Tricyclic compounds as TXA.sub.2 antagonists Tricyclic compounds as TXA.sub.2 antagonists

1992-11-23

1994-04-12

Raymond, Richard L.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

514245, 514246, 514248, 514249, 514258, 514299, 514300, 514301, 514302, 514303, 544180, 544211, 544212, 544219, 544235, 544236, 544253, 544264, 544278, 544280, 544349, 544350, 546112, 546113, 546114, 546115, 546117, 546118, A61K 31435, A61K 31505, C07D47104, C07D47300

Patent

active

053025962

ABSTRACT:
Novel tricyclic compound represented by formula ##STR1## possess a TXA.sub.2 biosynthesis inhibiting activity and/or a TXA.sub.2 receptor antagonizing activity, and are expected to have preventive and therapeutic effects on ischemic diseases, cerebro-vascular diseases, etc.

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